SCHEMBL24968162

SCHEMBL24968162

Cn1ncc2c(=O)[nH]ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
ERCC1 P07992 1/20 0.38
ERCC4 Q92889 1/20 0.38
PARP1 P09874 4/20 0.37
LMNA P02545 2/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
RAB9A P51151 1/20 0.34
BLM P54132 1/20 0.34
PARP15 Q460N3 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19434558 0.78 CNR1 (0.40) ALDH1A1BRD4KDM4EPRKACAPRKACG
SCHEMBL31318913 0.78 ALDH1A1 (0.35) ALDH1A1ERCC1ERCC4CCR4
SCHEMBL24035855 0.77 ALDH1A1 (0.36) ALDH1A1PARP1LMNAHPGDMAPK1
SCHEMBL13787655 0.72 ALDH1A1 (0.43) ALDH1A1ERCC1ERCC4PARP1LMNA
SCHEMBL31564540 0.71 MAPT (0.36) ALDH1A1PARP1CYP3A4CYP2C9RAB9A
SCHEMBL23047007 0.71 SMN1; SMN2 (0.51) ALDH1A1LMNAHPGDMAPK1HTT
SCHEMBL20551376 0.70 ALDH1A1 (0.42) ALDH1A1LMNAHPGDMAPK1HTT
SCHEMBL19154269 0.70 ALDH1A1 (0.39) ALDH1A1ERCC1ERCC4PARP1LMNA
SCHEMBL31564680 0.69 PARP1 (0.38) ALDH1A1PARP1LMNAHPGDKDM4E
SCHEMBL6800237 0.69 BRD4 (0.43) ALDH1A1PARP1LMNAHPGDBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4444305-A2 PHARMACEUTICAL COMPOUND Duke Street Bio Limited (GB) 2024-10-16 EP disclosed
WO-2023156386-A2 PHARMACEUTICAL COMPOUND Duke Street Bio Limited (GB) 2023-08-24 WO disclosed
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed