SCHEMBL24968488

SCHEMBL24968488

CC(C)(C)OC(=O)Nc1ccc(O[Si](C)(C)C(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 1/20 0.50
NAMPT P43490 1/20 0.50
CYP17A1 P05093 3/20 0.49
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA9 Q16790 1/20 0.44
LIPE Q05469 1/20 0.44
MAP4K4 O95819 1/20 0.43
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
MAPK14 Q16539 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GLS O94925 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159855 0.83 CYP17A1 (0.46) NAMPTCYP17A1CA12CA1CA9
SCHEMBL16476541 0.83 KMT2A (0.56) CA12CA1CA9
SCHEMBL13055402 0.82 CYP17A1 (0.59) PSMB8NAMPTCYP17A1CA12CA1
SCHEMBL22568337 0.81 CYP17A1 (0.46) PSMB8NAMPTCYP17A1CA12CA1
SCHEMBL17576495 0.81 CYP17A1 (0.48) PSMB8NAMPTCYP17A1CA12CA1
SCHEMBL29131710 0.80 HPGD (0.59) PSMB8NAMPTCYP17A1CA12CA1
SCHEMBL22581745 0.80 FAAH (0.56)
SCHEMBL17222455 0.80 NPC1 (0.58) NAMPTHDAC3HDAC8HDAC6
SCHEMBL1342005 0.79 SMN1; SMN2 (0.61) CYP17A1
SCHEMBL12085977 0.79 CYP17A1 (0.51) PSMB8NAMPTCYP17A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230115350-A1 TEAD INHIBITORS AND USES THEREOF CEDILLA THERAPEUTICS, INC. 2023-04-13 US disclosed
WO-2023009785-A1 TEAD INHIBITORS AND USES THEREOF CEDILLA THERAPEUTICS, INC. (US) 2023-02-02 WO disclosed
WO-2023009785-A1 TEAD INHIBITORS AND USES THEREOF CEDILLA THERAPEUTICS, INC. (US) 2023-02-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230115350-A1 TEAD INHIBITORS AND USES THEREOF TEAD2, TEAD3, TEAD4 PSMB8 3452/4885NAMPT 78/4885CYP17A1 1842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.