SCHEMBL24970949

SCHEMBL24970949

C=C(CC(C)(C)C)N1CCN(c2nc3cccnc3cc2Cl)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.40
HTR3B O95264 4/20 0.39
HTR3A P46098 4/20 0.39
TRPA1 O75762 3/20 0.39
HTR3E A5X5Y0 3/20 0.39
HTR3D Q70Z44 3/20 0.39
HTR3C Q8WXA8 3/20 0.39
KCNH2 Q12809 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
PHGDH O43175 1/20 0.37
HTR1A P08908 2/20 0.37
HRH4 Q9H3N8 1/20 0.37
SMO Q99835 2/20 0.37
GRM2 Q14416 1/20 0.36
CNR2 P34972 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30903372 0.79 POLB (0.55) TRPV1HTR3BHTR3ATRPA1HTR3E
SCHEMBL24970948 0.79 POLB (0.55) TRPV1HTR3BHTR3ATRPA1HTR3E
SCHEMBL24969735 0.75 KDM4E (0.52) HTR3BHTR3AHRH4
SCHEMBL24970163 0.75 TRPV1 (0.34) TRPV1TRPA1KCNH2TRPM8CNR2
SCHEMBL24970855 0.74 ALDH1A1 (0.43) HTR1AHRH4
SCHEMBL24971005 0.74 MEN1 (0.46) TRPV1PHGDHSMO
SCHEMBL24969955 0.73 HTR2C (0.52) HTR3BHTR3AHTR3EHTR3DHTR3C
SCHEMBL31142978 0.73 HTR2C (0.52) HTR3BHTR3AHTR3EHTR3DHTR3C
SCHEMBL24970110 0.73 KMT2A (0.43) TRPV1PHGDH
SCHEMBL24969924 0.72 TRPV1 (0.31) TRPV1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed