SCHEMBL24969735

SCHEMBL24969735

C=C(CC(C)(C)C)N1CCN(c2nc3ccccc3nc2CC)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.52
NPSR1 Q6W5P4 2/20 0.52
PKM P14618 1/20 0.52
RXFP1 Q9HBX9 3/20 0.48
MAPT P10636 2/20 0.48
HRH4 Q9H3N8 6/20 0.46
HRH1 P35367 1/20 0.45
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CSNK1A1 P48729 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24970855 0.79 ALDH1A1 (0.43) KDM4ENPSR1RXFP1MAPTHRH4
SCHEMBL29268329 0.77 HRH4 (0.71) KDM4ENPSR1PKMRXFP1MAPT
SCHEMBL24970949 0.75 TRPV1 (0.40) HRH4HTR3BHTR3A
SCHEMBL7237642 0.73 KDM4E (0.58) KDM4ENPSR1PKMRXFP1MAPT
SCHEMBL24951560 0.68 GBA1 (0.53)
SCHEMBL31133544 0.68 GBA1 (0.53)
SCHEMBL24970904 0.67 MEN1 (0.45) NPSR1MAPTALDH1A1
SCHEMBL24970163 0.66 TRPV1 (0.34) KDM4EMAPTALDH1A1TSHRMAPK1
SCHEMBL21163168 0.66 GPR119 (0.47)
SCHEMBL22936027 0.66 PHGDH (0.40) KDM4EHRH4ALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed