SCHEMBL24970965

SCHEMBL24970965

Cc1c(Cl)ccc2cc(Cl)c(=O)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.49
DAO P14920 3/20 0.42
GRIN2D O15399 5/20 0.41
GRIN3B O60391 5/20 0.41
GRIN1 Q05586 5/20 0.41
GRIN2A Q12879 5/20 0.41
GRIN2B Q13224 5/20 0.41
GRIN2C Q14957 5/20 0.41
GRIN3A Q8TCU5 5/20 0.41
HSD17B10 Q99714 6/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TSHR P16473 2/20 0.38
DDO Q99489 1/20 0.38
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31143052 1.00 MAPT (0.49) MAPTDAOGRIN2DGRIN3BGRIN1
SCHEMBL3360987 0.84 DAO (0.61) MAPTDAODDO
SCHEMBL24970979 0.76 DAO (0.65) DAOHSD17B10KDM4EALDH1A1HPGD
SCHEMBL29955876 0.75 MAPT (0.46) MAPTDAOALDH1A1CSNK2A2CSNK2B
SCHEMBL3605104 0.74 HPGD (0.53) MAPTDAOHSD17B10KDM4EALDH1A1
SCHEMBL28881409 0.70 DAO (0.64) MAPTDAOHSD17B10KDM4EALDH1A1
SCHEMBL30235048 0.70 DAO (0.38) MAPTDAOGRIN2DGRIN3BGRIN1
SCHEMBL25604921 0.70 DAO (0.38) MAPTDAOGRIN2DGRIN3BGRIN1
SCHEMBL4048527 0.68 CDK1 (0.64) MAPTHSD17B10KDM4EALDH1A1HPGD
SCHEMBL25418850 0.68 TDP1 (0.37) DAOGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed