SCHEMBL24971015

SCHEMBL24971015

Cc1c(Cl)ccc2cc(Cl)c(Cl)nc12

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.36
MAPT P10636 3/20 0.35
CCR1 P32246 3/20 0.34
CCR8 P51685 2/20 0.34
CCR5 P51681 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 4/20 0.33
NPSR1 Q6W5P4 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PDPK1 O15530 1/20 0.31
NPC1 O15118 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPK1 P28482 1/20 0.31
NR4A2 P43354 1/20 0.30
KMT2A Q03164 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31143096 1.00 PPARA (0.36) PPARAMAPTCCR1CCR8CCR5
SCHEMBL9730937 0.86 ALDH1A1 (0.35) PPARAMAPTCCR1CCR8CCR5
SCHEMBL3877857 0.78 MEN1 (0.35) PPARAMAPTCCR1CCR8CCR5
SCHEMBL31490208 0.74 CCR1 (0.61) MAPTCCR1CCR5L3MBTL1KDM4E
SCHEMBL9186312 0.74 CCR1 (0.61) MAPTCCR1CCR5L3MBTL1KDM4E
SCHEMBL31142923 0.73 DRD4 (0.51) MAPTL3MBTL1ALDH1A1NPC1KDM4E
SCHEMBL24971012 0.73 DRD4 (0.51) MAPTL3MBTL1ALDH1A1NPC1KDM4E
SCHEMBL7025162 0.72 CCR1 (0.45) PPARAMAPTCCR1CCR8CCR5
SCHEMBL6888604 0.72 CCR1 (0.67) PPARAMAPTCCR1CCR8CCR5
SCHEMBL29890061 0.72 CCR1 (0.67) PPARAMAPTCCR1CCR8CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed