SCHEMBL9730937

SCHEMBL9730937

Cc1cc2ccc(Cl)c(C)c2nc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
PPARA Q07869 1/20 0.35
MAPT P10636 3/20 0.34
CCR1 P32246 2/20 0.33
CCR8 P51685 2/20 0.33
CCR5 P51681 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
PDPK1 O15530 1/20 0.31
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410188 0.86 MEN1 (0.46) ALDH1A1MEN1TSHRKMT2AMAPT
SCHEMBL24971015 0.86 PPARA (0.36) ALDH1A1KMT2APPARAMAPTCCR1
SCHEMBL31143096 0.86 PPARA (0.36) ALDH1A1KMT2APPARAMAPTCCR1
SCHEMBL3877857 0.84 MEN1 (0.35) MEN1TSHRKMT2APPARAMAPT
SCHEMBL9732163 0.73 DRD4 (0.53) MEN1KMT2AMAPTKDM4EMAPK1
SCHEMBL18289967 0.73 L3MBTL1 (0.53) ALDH1A1TSHRKMT2AMAPTCCR1
SCHEMBL31490208 0.72 CCR1 (0.61) KMT2AMAPTCCR1CCR5KDM4E
SCHEMBL9186312 0.72 CCR1 (0.61) KMT2AMAPTCCR1CCR5KDM4E
SCHEMBL7025162 0.71 CCR1 (0.45) MEN1TSHRKMT2APPARAMAPT
SCHEMBL6888604 0.71 CCR1 (0.67) PPARAMAPTCCR1CCR8CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5104884-A Rheumatic diseases, fungicides ALKALOIDA VEGYESZETI GYAR (HU) 1992-04-14 US disclosed
EP-0221947-B1 TRIAZOLYL QUINOLINE DERIVATIVES ALKALOIDA VEGYéSZETI GYáR (HU) 1990-11-28 EP disclosed
EP-0221947-A1 TRIAZOLYL QUINOLINE DERIVATIVES. ALKALOIDA VEGYESZETI GYAR (HU) 1987-05-20 EP disclosed
WO-1986006721-A1 TRIAZOLYL QUINOLINE DERIVATIVES ALKALOIDA VEGYÉSZETI GYÁR (HU) 1986-11-20 WO disclosed