SCHEMBL24975658

SCHEMBL24975658

CC(=O)c1ccc2nc(C)cc(-c3cccc(C(=O)OC(C)(C)C)c3)c2c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
DHFR P00374 2/20 0.43
TP53 P04637 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
ABCB1 P08183 1/20 0.42
GUSB P08236 1/20 0.41
MAPT P10636 1/20 0.41
SLC7A5 Q01650 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 2/20 0.41
HTT P42858 2/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MMP1 P03956 2/20 0.39
MMP9 P14780 2/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24976143 0.90 ABCG2 (0.46) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL31428903 0.90 ABCG2 (0.46) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL24975655 0.89 LMNA (0.44) NPC1TP53ABCG2GUSBMAPT
SCHEMBL24975485 0.87 ABCG2 (0.47) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL31428518 0.87 ABCG2 (0.47) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL31428407 0.84 ABCG2 (0.43) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL24975465 0.84 ABCG2 (0.43) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL31428875 0.84 ABCG2 (0.49) NPC1TP53ABCG2ABCB1GUSB
SCHEMBL31428552 0.84 MEN1 (0.46) KDM4EMEN1KMT2AL3MBTL1
SCHEMBL24976140 0.81 TP53 (0.46) NPC1TP53ABCG2ABCB1GUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023008577-A1 RAS/RAF BINDING INHIBITOR COMPOUND 国立大学法人神戸大学 2023-02-02 WO disclosed