SCHEMBL249761

SCHEMBL249761

CCCCCOc1ccc(S(=O)(=O)O)c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.54
FABP4 P15090 6/20 0.54
FABP5 Q01469 6/20 0.54
CNR1 P21554 3/20 0.53
CNR2 P34972 3/20 0.53
CYP2C9 P11712 1/20 0.53
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
HTT P42858 2/20 0.49
S1PR3 Q99500 1/20 0.48
GAA P10253 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TSHR P16473 2/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225810 0.97 SLC2A1 (0.55) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL11337934 0.89 SLC2A1 (0.48) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL11337933 0.89 SLC2A1 (0.48) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL22738512 0.89 SLC2A1 (0.53) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL13812467 0.84 TSHR (0.59) SLC2A1FABP4MEN1KMT2ATHRB
SCHEMBL9124215 0.84 FABP4 (0.52) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL9124205 0.84 FABP4 (0.52) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL23649347 0.84 MEN1 (0.43) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL11239189 0.83 S1PR3 (0.47) SLC2A1FABP4FABP5CNR1CNR2
SCHEMBL10907588 0.83 FABP4 (0.52) SLC2A1FABP4FABP5CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339663-B1 NAPHTHALENE DERIVATIVES NOVARTIS AG (CH) 2012-01-04 EP disclosed
EP-2338886-A2 Naphthalene derivatives Novartis AG (CH) 2011-06-29 EP disclosed
US-7045533-B2 Such as naphthalen-1-yl-(4-pentyloxy-naphthalen-1-yl)-mehtane for treatment/prevention of diseases/conditions associated with cannobinoid receptor activation such as chronic pain, osteo- and rheumatoid arthritis, teno-synovitis and gout NOVARTIS AG (CH) 2006-05-16 US disclosed
CN-1224598-C Naphthalene derivatives NOVARTIS AG (CH) 2005-10-26 CN disclosed
US-20040053890-A1 Naphthalene derivatives NOVARTIS AG (CH) 2004-03-18 US disclosed
CN-1476424-A Naphthalene derivatives ��˹��ŵ�� 2004-02-18 CN disclosed
EP-1339663-A2 NAPHTHALENE DERIVATIVES Novartis AG (CH) 2003-09-03 EP disclosed
WO-2002042248-A2 NAPHTHALENE DERIVATIVES NOVARTIS AG (CH) 2002-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053890-A1 Naphthalene derivatives CYP1A1, SULT1E1, CYP2F1 SLC2A1 4319/4885FABP4 4291/4885FABP5 3822/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.