SCHEMBL24980488

SCHEMBL24980488

CCCn1cnc2c(N)nc(F)nc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.60
ADORA1 P30542 5/20 0.60
ADORA2B P29275 2/20 0.60
TMIGD3 P0DMS9 3/20 0.55
CDK1 P06493 2/20 0.54
CCNB1 P14635 2/20 0.54
CCNE1 P24864 2/20 0.54
CDK2 P24941 2/20 0.54
CYP2C19 P33261 2/20 0.46
PI4KA P42356 1/20 0.44
PI4K2B Q8TCG2 1/20 0.44
PI4K2A Q9BTU6 1/20 0.44
PI4KB Q9UBF8 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HIF1A Q16665 1/20 0.43
AHCY P23526 2/20 0.43
SLC29A1 Q99808 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21451434 0.87 CDK1 (0.71) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL1377647 0.84 CDK1 (0.76) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL232387 0.83 ADORA2A (0.62) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL3441081 0.81 CDK1 (0.64) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL19553561 0.81 ADORA2A (0.57) ADORA2AADORA1CDK1CCNB1CCNE1
SCHEMBL21128125 0.81 CDK1 (0.50) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL28476413 0.79 ADORA2A (0.57) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL23350293 0.78 ALDH1A1 (0.44) ADORA2AADORA1ADORA2BTMIGD3CDK1
SCHEMBL130527 0.78 CDK1 (0.64) ADORA2AADORA1ADORA2BCDK1CCNB1
SCHEMBL21504451 0.78 CCNE1 (0.46) ADORA2AADORA1CDK1CCNB1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023000708-A1 POLYSUBSTITUTED PURINE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2023-01-26 WO disclosed
WO-2023000708-A1 POLYSUBSTITUTED PURINE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2023-01-26 WO disclosed
CN-113549076-A Polysubstituted purine compound and preparation method and application thereof 中国药科大学 2021-10-26 CN disclosed