SCHEMBL2498448

SCHEMBL2498448

NCC(=O)c1ccc2n1CCc1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.37
HDAC1 Q13547 1/20 0.36
MTNR1A P48039 4/20 0.36
MTNR1B P49286 4/20 0.36
GPR84 Q9NQS5 1/20 0.35
TSHR P16473 3/20 0.35
SRD5A1 P18405 1/20 0.35
SRD5A2 P31213 1/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PTAFR P25105 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC6A2 P23975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1158808 0.84 BCAT2 (0.46) BCAT2HDAC1MTNR1AMTNR1BGPR84
SCHEMBL31105304 0.82 SRD5A1 (0.41) BCAT2HDAC1MTNR1AMTNR1BTSHR
SCHEMBL2517925 0.81 MTNR1A (0.41) HDAC1MTNR1AMTNR1BMAPTMEN1
SCHEMBL1159546 0.77 AKT1 (0.35) BCAT2HDAC1MTNR1AMTNR1BGPR84
SCHEMBL2736494 0.71 CES1 (0.41) BCAT2GPR84TSHRMAPTSMN1; SMN2
SCHEMBL215395 0.70 SERPINE1 (0.39) BCAT2GPR84TSHRSRD5A1SRD5A2
SCHEMBL2778467 0.69 HRH1 (0.43) BCAT2HDAC1GPR84MAPTSMN1; SMN2
SCHEMBL3395760 0.68 KDM4E (0.39) HDAC1MTNR1AMTNR1BGPR84MAPT
SCHEMBL5658471 0.67 CES1 (0.44) BCAT2GPR84MAPTSMN1; SMN2KDM4E
SCHEMBL3397210 0.67 HDAC1 (0.48) HDAC1MTNR1AMTNR1BTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252611-B1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES ORGANON NV (NL) 2011-10-05 EP disclosed