SCHEMBL25002889

SCHEMBL25002889

COC(=O)c1ccc(-c2ccc(OC(C)C)cc2)o1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.51
POLB P06746 2/20 0.47
KMT2A Q03164 4/20 0.46
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
ATM Q13315 1/20 0.46
SCN10A Q9Y5Y9 2/20 0.46
HTT P42858 1/20 0.45
ERCC5 P28715 1/20 0.45
FEN1 P39748 1/20 0.45
SETD7 Q8WTS6 1/20 0.44
ALDH1A1 P00352 3/20 0.44
THRB P10828 1/20 0.44
HTR1A P08908 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CNR1 P21554 1/20 0.44
DRD1 P21728 1/20 0.44
HTR2A P28223 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25003808 0.84 ABCB1 (0.48) ABCB1POLBKMT2AMAPTMEN1
SCHEMBL4943612 0.84 ALDH1A1 (0.57) POLBKMT2AMAPTMEN1CYP1A2
SCHEMBL4943742 0.79 HTT (0.51) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL21981938 0.78 HTT (0.67) POLBKMT2AMAPTMEN1CYP1A2
SCHEMBL1143497 0.78 ALDH1A1 (0.50) POLBKMT2AMAPTMEN1CYP1A2
SCHEMBL22066403 0.78 HPGD (0.56) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL4946307 0.78 LMNA (0.57) POLBKMT2AMAPTMEN1CYP1A2
SCHEMBL25002899 0.78 ALDH1A1 (0.65) MAPTSCN10AERCC5FEN1ALDH1A1
SCHEMBL3059132 0.77 ALDH1A1 (0.62) POLBKMT2AMEN1CYP1A2CYP2C19
SCHEMBL26263255 0.77 SUCNR1 (0.64) ERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023010192-A1 N-ACYLHYDRAZONE COMPOUNDS CAPABLE OF INHIBITING NAV1.7 AND/OR NAV1.8, PROCESSES FOR THE PREPARATION THEREOF, COMPOSITIONS, USES, METHODS FOR TREATMENT USING SAME, AND KITS EUROFARMA LABORATÓRIOS S.A. (BR) 2023-02-09 WO disclosed