SCHEMBL25003989

SCHEMBL25003989

Cc1cccc(N2CCN(CCCCOc3ccc4c(c3)NC(O)C3CC43)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.52
DRD2 P14416 5/20 0.48
HTR1A P08908 4/20 0.44
HTR2A P28223 3/20 0.44
DRD3 P35462 3/20 0.44
HTR2C P28335 2/20 0.44
HTR7 P34969 2/20 0.43
ADRA1A P35348 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25003992 0.86 DRD2 (0.59) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003629 0.84 DRD2 (0.51) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003004 0.84 DRD2 (0.56) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL30839786 0.83 DRD2 (0.55) KCNH2DRD2HTR7
SCHEMBL25003003 0.83 DRD2 (0.55) KCNH2DRD2HTR7
SCHEMBL25003854 0.83 KCNH2 (0.53) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003035 0.82 DRD2 (0.59) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003853 0.82 DRD2 (0.59) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003011 0.81 DRD2 (0.49) KCNH2DRD2HTR1AHTR2ADRD3
SCHEMBL25003990 0.79 DRD2 (0.49) KCNH2DRD2HTR1AHTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011608-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海枢境生物科技有限公司 2023-02-09 WO disclosed