SCHEMBL25003992

SCHEMBL25003992

Cc1cccc(N2CCN(CCCCOc3ccc4c(c3)NC(O)C3CC43)CC2)c1C

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.59
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
DRD3 P35462 2/20 0.44
HTR1A P08908 2/20 0.44
HTR2A P28223 2/20 0.44
KCNH2 Q12809 1/20 0.44
DRD4 P21917 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25003629 0.91 DRD2 (0.51) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003004 0.88 DRD2 (0.56) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003035 0.86 DRD2 (0.59) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003853 0.86 DRD2 (0.59) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003989 0.86 KCNH2 (0.52) DRD2DRD3HTR1AHTR2AKCNH2
SCHEMBL25003011 0.85 DRD2 (0.49) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003990 0.82 DRD2 (0.49) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003982 0.82 DRD2 (0.58) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003041 0.82 DRD2 (0.68) DRD2MAPTDRD3HTR1AHTR2A
SCHEMBL25003061 0.81 DRD2 (0.58) DRD2MAPTDRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011608-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海枢境生物科技有限公司 2023-02-09 WO disclosed