SCHEMBL2501207

SCHEMBL2501207

COC(=O)C[C@H](O[Si](C(C)C)(C(C)C)C(C)C)[C@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
ELANE P08246 2/20 0.45
CTSK P43235 4/20 0.43
CTSL P07711 3/20 0.43
CTSS P25774 3/20 0.43
CTSB P07858 2/20 0.43
PRTN3 P24158 1/20 0.43
REN P00797 1/20 0.42
ABCB1 P08183 1/20 0.42
TOP2A P11388 1/20 0.42
TOP2B Q02880 1/20 0.42
CTRB1 P17538 2/20 0.42
CAPN1 P07384 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2492793 0.91 ATM (0.49) ATMELANECTSKCTSLCTSS
SCHEMBL14493005 0.83 ATM (0.39) ATMELANECTSKCTSLCTSS
SCHEMBL2493028 0.81 ABCB1 (0.54) ATMELANECTSKCTSLCTSS
SCHEMBL12906609 0.79 ATM (0.61) ATMELANECTSKCTSLCTSS
SCHEMBL2392482 0.78 ATM (0.46) ATMELANECTSKCTSLCTSS
SCHEMBL9937088 0.77 TRPM8 (0.55) ATMELANECTSKCTSLCTSS
SCHEMBL9937089 0.77 TRPM8 (0.55) ATMELANECTSKCTSLCTSS
SCHEMBL3276084 0.77 ATM (0.49) ATMELANECTSKCTSLCTSS
SCHEMBL6841182 0.77 ATM (0.56) ATMELANECTSKCTSLCTSS
SCHEMBL8972716 0.77 ATM (0.56) ATMELANECTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030279-B2 Tamandarin analogs and fragments thereof and methods of making and using THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2011-10-04 US disclosed
US-20070149446-A1 Tamandarin analogs and fragments thereof and methods of making and using THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA CENTER FOR TECHNOLOGY TRANSFER (US) 2007-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149446-A1 Tamandarin analogs and fragments thereof and methods of making and using FOXM1, F3, RB1 ATM 1572/4885ELANE 1539/4885CTSK 353/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.