SCHEMBL25023217

SCHEMBL25023217

COC(=O)[C@H]1CNC(=O)CN1C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 0.44
ANPEP P15144 4/20 0.44
BRD4 O60885 1/20 0.41
CYP1A2 P05177 1/20 0.36
HIF1A Q16665 1/20 0.36
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
FKBP1A P62942 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CYP19A1 P11511 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14826526 1.00 MMP2 (0.44) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL14826522 0.80 TSHR (0.34)
SCHEMBL30191457 0.77 P2RX7 (0.46) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL8231723 0.77 P2RX7 (0.46) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL1637512 0.77 P2RX7 (0.46) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL17973099 0.77 MMP2 (0.60) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL13403397 0.77 MMP2 (0.60) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL2691165 0.77 MMP2 (0.60) MMP2ANPEPBRD4CYP1A2HIF1A
SCHEMBL31749294 0.74 PTPN1 (0.46) MMP2ANPEP
SCHEMBL13567829 0.74 PTPN1 (0.46) MMP2ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240156780-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF AXIAL THERAPEUTICS, INC. (US) 2024-05-16 US disclosed
US-11951094-B2 TLR2 modulator compounds, pharmaceutical compositions and uses thereof AXIAL THERAPEUTICS, INC. (US) 2024-04-09 US disclosed
EP-4171547-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Axial Therapeutics, Inc. (US) 2023-05-03 EP disclosed
US-20230051773-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF AXIAL THERAPEUTICS, INC. (US) 2023-02-16 US disclosed
US-20230051773-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF AXIAL THERAPEUTICS, INC. (US) 2023-02-16 US disclosed
CN-115666553-A TLR2 modulator compounds, and pharmaceutical compositions and uses thereof 轴向治疗公司 2023-01-31 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230051773-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF TLR2, TLR3, TLR4 MMP2 1506/4885ANPEP 3602/4885BRD4 765/4885
US-20240156780-A1 TLR2 MODULATOR COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF TLR2, TLR3, TLR4 MMP2 1506/4885ANPEP 3602/4885BRD4 765/4885
US-11951094-B2 TLR2 modulator compounds, pharmaceutical compositions and uses thereof TLR2, TLR3, TLR4 MMP2 1506/4885ANPEP 3602/4885BRD4 765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.