SCHEMBL25028087

SCHEMBL25028087

c1ccc(N(c2ccncc2)c2ccc3c4cccc5cccc(c6cccc2c63)c54)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
THRB P10828 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ERBB2 P04626 1/20 0.34
FYN P06241 1/20 0.34
MAOA P21397 1/20 0.34
ACHE P22303 1/20 0.34
AHR P35869 1/20 0.34
SLC6A2 P23975 4/20 0.33
SIGMAR1 Q99720 2/20 0.33
KDM1A O60341 1/20 0.32
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25028133 0.95 CYP1A2 (0.35) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL4026976 0.91 ALDH1A1 (0.43) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL13899997 0.89 ALDH1A1 (0.42) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL13320967 0.87 ALDH1A1 (0.34) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL13320974 0.87 ALDH1A1 (0.34) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL25027804 0.87 ALDH1A1 (0.37) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL25027743 0.84 SIGMAR1 (0.44) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL13899996 0.84 CYP1A2 (0.38) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL14262670 0.84 CYP1A2 (0.40) CYP1A2ALDH1A1HPGDTHRBHSD17B10
SCHEMBL13320952 0.84 CYP1A2 (0.50) CYP1A2ALDH1A1HPGDTHRBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230050869-A1 THERMOELECTRIC CONVERSION MATERIAL, AND THERMOELECTRIC CONVERSION ELEMENT PREPARED THEREWITH TOYO INK SC HOLDINGS CO., LTD. (JP) 2023-02-16 US disclosed