SCHEMBL2503145

SCHEMBL2503145

NC(=O)C1CCN(C(=O)O)C1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
KDM4E B2RXH2 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GLA P06280 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28774060 0.88 ALDH1A1 (0.57) GAAKDM4EALDH1A1MAPK1LMNA
SCHEMBL25363482 0.88 ALDH1A1 (0.57) GAAKDM4EALDH1A1MAPK1LMNA
SCHEMBL2224391 0.88 ALDH1A1 (0.57) GAAKDM4EALDH1A1MAPK1LMNA
SCHEMBL2030080 0.86 GAA (0.55) GAAKDM4ESMN1; SMN2ALDH1A1TDP1
SCHEMBL30793930 0.86 ALDH1A1 (0.51) KDM4ESMN1; SMN2ALDH1A1MAPK1LMNA
SCHEMBL3938968 0.84 GAA (0.48) GAAKDM4ESMN1; SMN2ALDH1A1MAPK1
SCHEMBL15376451 0.83 SMN1; SMN2 (0.40) GAAKDM4ESMN1; SMN2ALDH1A1MAPK1
SCHEMBL2875954 0.82 NOTUM (0.46) ALDH1A1LMNA
SCHEMBL652433 0.82 NOTUM (0.46) ALDH1A1LMNA
SCHEMBL2875175 0.82 NOTUM (0.46) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3365339-A1 NOVEL FERROPORTIN INHIBITORS Vifor (International) AG (CH) 2018-08-29 EP disclosed
WO-2017068090-A1 NOVEL FERROPORTIN INHIBITORS VIFOR (INTERNATIONAL) AG (CH) 2017-04-27 WO disclosed
EP-2375904-B1 BIARYL CARBOXAMIDES MERCK SHARP & DOHME (US) 2014-05-28 EP disclosed
EP-2375904-A1 BIARYL CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2011-10-19 EP disclosed
WO-2010077624-A1 BIARYL CARBOXAMIDES MERCK SHARP & DOHME CORP. (US) 2010-07-08 WO disclosed