SCHEMBL2875175

SCHEMBL2875175

O=C(O)[C@@H]1CCN(C(=O)O)C1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 9/20 0.46
LMNA P02545 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652433 1.00 NOTUM (0.46) NOTUMLMNAL3MBTL1MAPTRAB9A
SCHEMBL2875954 1.00 NOTUM (0.46) NOTUMLMNAL3MBTL1MAPTRAB9A
SCHEMBL2878783 0.86 ALDH1A1 (0.49) MAPTALDH1A1
SCHEMBL316646 0.86 ALDH1A1 (0.49) MAPTALDH1A1
SCHEMBL2880648 0.86 ALDH1A1 (0.49) MAPTALDH1A1
SCHEMBL28026037 0.86 NOTUM (0.46) NOTUMLMNAL3MBTL1MAPTRAB9A
SCHEMBL587681 0.85 LMNA (0.53) LMNAL3MBTL1MAPTRAB9APOLB
Bromide SCHEMBL3964464 0.85 ALDH1A1 (0.47) MAPTALDH1A1
SCHEMBL7357706 0.85 ALDH1A1 (0.48) LMNAPOLBALDH1A1
SCHEMBL25317162 0.82 LMNA (0.39) LMNAPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023240038-A1 TRICYCLIC QUINOLONE BCL6 BIFUNCTIONAL DEGRADERS Treeline Biosciences, Inc. (US) 2023-12-14 WO disclosed
WO-2023086399-A1 BIFUNCTIONAL DEGRADERS OF HEMATOPOIETIC PROGENITOR KINASE AND THERAPEUTIC USES THEREOF NURIX THERAPEUTICS, INC. (US) 2023-05-19 WO disclosed
WO-2023086341-A1 INHIBITORS OF KRAS BIOMEA FUSION, INC. (US) 2023-05-19 WO disclosed
US-8410100-B2 Pteridinone derivatives as PI3-kinases inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-04-02 US disclosed
EP-2114945-B1 PTERIDINONE DERIVATIVES AS PI3-KINASES INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2010-10-20 EP disclosed
US-20100099680-A1 PTERIDINONE DERIVATIVES AS P13-KINASES INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-22 US disclosed
EP-2114945-A1 PTERIDINONE DERIVATIVES AS PI3-KINASES INHIBITORS Boehringer Ingelheim International GmbH (DE) 2009-11-11 EP disclosed
WO-2008092831-A1 PTERIDINONE DERIVATIVES AS PI3-KINASES INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-07 WO disclosed
EP-1953163-A1 Pteridinone derivatives as PI3-kinases inhibitors Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2008-08-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100099680-A1 PTERIDINONE DERIVATIVES AS P13-KINASES INHIBITORS PIK3CA, PDPK1, PIK3C3 NOTUM 3199/4885LMNA 3269/4885L3MBTL1 4578/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.