SCHEMBL25044792

SCHEMBL25044792

Cc1nnn(-c2ccc(C(F)(F)F)cc2)c1COc1ccc(Cl)nn1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 11/20 0.43
GABRB3 P28472 10/20 0.43
GABRG2 P18507 8/20 0.43
KCNH2 Q12809 4/20 0.43
BRAF P15056 1/20 0.35
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RXRA P19793 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30282901 0.87 GABRA5 (0.54) GABRA5GABRB3GABRG2KCNH2
SCHEMBL25045396 0.87 GABRA5 (0.44) GABRA5GABRB3GABRG2KCNH2
SCHEMBL25044752 0.87 GABRA5 (0.44) GABRA5GABRB3GABRG2KCNH2L3MBTL1
SCHEMBL30283019 0.85 GABRA5 (0.43) GABRA5GABRB3GABRG2KCNH2
SCHEMBL25045401 0.85 GABRA5 (0.43) GABRA5GABRB3GABRG2KCNH2
SCHEMBL30236918 0.84 GABRA5 (0.41) GABRA5GABRB3GABRG2KCNH2RAB9A
SCHEMBL21623964 0.84 GABRA5 (0.43) GABRA5GABRB3GABRG2KCNH2RXRA
SCHEMBL30282856 0.84 GABRA5 (0.43) GABRA5GABRB3GABRG2KCNH2RXRA
SCHEMBL25045127 0.83 GABRA5 (0.41) GABRA5GABRB3GABRG2KCNH2
SCHEMBL25045399 0.83 GABRA5 (0.43) GABRA5GABRB3GABRG2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023016521-A1 SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 上海赛默罗生物科技有限公司 2023-02-16 WO disclosed