SCHEMBL25051768

SCHEMBL25051768

Bc1ccc(F)c2sc(NC(=O)OC(C)(C)C)c(C#N)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
TRPA1 O75762 1/20 0.35
EGLN2 Q96KS0 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
CTSS P25774 3/20 0.32
CTSK P43235 3/20 0.32
CYP17A1 P05093 1/20 0.32
ALDH1A1 P00352 5/20 0.32
NPC1 O15118 4/20 0.32
RAB9A P51151 4/20 0.32
MAPT P10636 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23498289 0.87 MEN1 (0.36) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL29812974 0.87 MEN1 (0.36) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL24917988 0.86 MEN1 (0.35) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL25049486 0.83 CYP17A1 (0.33) CYP17A1PSMB8POLBLMNA
SCHEMBL30781872 0.80 TRPA1 (0.35) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL27100884 0.80 TRPA1 (0.35) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL31670679 0.80 MEN1 (0.36) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL30537698 0.80 MEN1 (0.32) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL24757043 0.80 AAK1 (0.33) MEN1KMT2ATRPA1EGLN2CYP1A2
SCHEMBL25405428 0.80 MEN1 (0.32) MEN1KMT2ATRPA1EGLN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023215801-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2023-11-09 WO disclosed
WO-2023098832-A1 PYRIDOPYRIMIDINE DERIVATIVES SERVING AS SMALL GTP ENZYME KRAS MUTATION INHIBITORS 思路迪生物医药(上海)有限公司 2023-06-08 WO disclosed
WO-2023018699-A1 SELECTIVE KRAS INHIBITORS ERASCA, INC. (US) 2023-02-16 WO disclosed