SCHEMBL25075368

SCHEMBL25075368

COC(=O)c1ccn(C[C@H](C)N)c(=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
POLB P06746 1/20 0.44
APOBEC3A P31941 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
HTR2C P28335 13/20 0.43
SLC7A5 Q01650 1/20 0.41
LOXL2 Q9Y4K0 2/20 0.40
MAPT P10636 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
ATM Q13315 1/20 0.39
HTR2A P28223 10/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29169174 1.00 KDM4E (0.44) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL1015082 0.88 ALDH1A1 (0.46) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL29168988 0.84 HTR2C (0.41) HSD17B10HTR2CHTR2A
SCHEMBL29168986 0.84 HTR2C (0.41) HSD17B10HTR2CHTR2A
SCHEMBL14527151 0.80 HTR2C (0.63) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL29169075 0.78 LMNA (0.56) KDM4EALDH1A1SMN1; SMN2LOXL2MAPT
SCHEMBL25075523 0.78 LMNA (0.56) KDM4EALDH1A1SMN1; SMN2LOXL2MAPT
SCHEMBL29168967 0.77 KDM4E (0.41) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL29168963 0.77 KDM4E (0.41) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL12180387 0.77 ALDH1A1 (0.48) KDM4EALDH1A1HPGDHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117377665-A PARP7 inhibitor and application thereof 北京华森英诺生物科技有限公司 2024-01-09 CN disclosed
WO-2023020479-A1 PARP7 INHIBITOR AND APPLICATION THEREOF 重庆华森制药股份有限公司 2023-02-23 WO disclosed