SCHEMBL25075372

SCHEMBL25075372

CCOC(=O)c1cccn(C[C@@H](C)O)c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
KDM4E B2RXH2 10/20 0.45
ALDH1A1 P00352 8/20 0.45
HPGD P15428 5/20 0.45
GAA P10253 4/20 0.45
GLA P06280 3/20 0.45
HSD17B10 Q99714 2/20 0.44
RXFP1 Q9HBX9 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.41
STAT6 P42226 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29168930 1.00 TSHR (0.50) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL25075378 0.86 TSHR (0.47) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL25075373 0.85 TSHR (0.43) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL29169172 0.85 TSHR (0.43) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL29169168 0.82 TSHR (0.43) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL29169165 0.82 TSHR (0.43) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL29169016 0.81 BRD4 (0.48) KDM4EALDH1A1HSD17B10MAPTBRD4
SCHEMBL29169021 0.81 BRD4 (0.48) KDM4EALDH1A1HSD17B10MAPTBRD4
SCHEMBL11639000 0.80 ALDH1A1 (0.54) TSHRKDM4EALDH1A1HPGDGAA
SCHEMBL20594715 0.78 TSHR (0.54) TSHRKDM4EALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117377665-A PARP7 inhibitor and application thereof 北京华森英诺生物科技有限公司 2024-01-09 CN disclosed
WO-2023020479-A1 PARP7 INHIBITOR AND APPLICATION THEREOF 重庆华森制药股份有限公司 2023-02-23 WO disclosed