SCHEMBL25079908

SCHEMBL25079908

N#Cc1n[nH]c2ccc(-c3ccc(SN4CCC(Nc5ccc(C(F)(F)F)cc5)CC4)cc3)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 5/20 0.38
WNT1 P04628 3/20 0.38
AXL P30530 1/20 0.36
HTR6 P50406 2/20 0.36
LRRK2 Q5S007 3/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
MAPK1 P28482 2/20 0.35
MAP2K4 P45985 2/20 0.35
MAPKAPK3 Q16644 2/20 0.35
MAPK6 Q16659 2/20 0.35
MAPKAPK2 P49137 1/20 0.35
PHGDH O43175 1/20 0.35
NTRK1 P04629 1/20 0.34
PAK1 Q13153 1/20 0.33
DHODH Q02127 1/20 0.33
CCR6 P51684 1/20 0.33
TEAD1 P28347 1/20 0.33
TEAD4 Q15561 1/20 0.33
TEAD2 Q15562 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25079791 0.89 CCR6 (0.44) DYRK1AWNT1CCR6
SCHEMBL25079907 0.83 CCR6 (0.52) HTR6CCR6
SCHEMBL25079510 0.78 MAP3K12 (0.42) DYRK1APAK1CCR6
SCHEMBL25079719 0.77 CCR6 (0.45) DYRK1AWNT1CCR6
SCHEMBL25079902 0.77 CCR6 (0.45) DYRK1AWNT1CCR6
SCHEMBL25079903 0.77 CCR6 (0.45) DYRK1AWNT1CCR6
SCHEMBL25079573 0.74 KIF11 (0.50)
SCHEMBL25079785 0.73 CCR6 (0.65) CCR6
SCHEMBL30284751 0.73 CCR6 (0.65) CCR6
SCHEMBL31155642 0.73 CCR6 (0.49) CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023023534-A2 ARYL SULFONYL COMPOUNDS AS CCR6 INHIBITORS CHEMOCENTRYX, INC. (US) 2023-02-23 WO disclosed