SCHEMBL25079573

SCHEMBL25079573

O=C1Cc2cc(-c3ccc(SN4CCC(Nc5ccc(C(F)(F)F)cc5)CC4)cc3)ccc2N1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.50
TDP2 O95551 1/20 0.44
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
GAA P10253 1/20 0.42
CDK2 P24941 2/20 0.42
AKT1 P31749 2/20 0.42
CDK1 P06493 1/20 0.42
KIT P10721 1/20 0.42
KDR P35968 1/20 0.42
GRIA1 P42261 4/20 0.39
MET P08581 1/20 0.39
PGR P06401 2/20 0.38
ULK1 O75385 1/20 0.38
SMYD3 Q9H7B4 1/20 0.37
PTK2B Q14289 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25079861 0.88 CCR6 (0.48) KIF11CDK2AKT1CDK1KIT
SCHEMBL25079568 0.82 GAA (0.60) KIF11GAACDK2SMYD3
SCHEMBL30284876 0.82 GAA (0.60) KIF11GAACDK2SMYD3
SCHEMBL25079839 0.81 CCR6 (0.48) CDK2
SCHEMBL25079308 0.79 CRBN (0.45) CDK2AKT1CDK1KITKDR
SCHEMBL1903306 0.77 KIF11 (0.80) KIF11TDP2PDE3BPDE3AGAA
SCHEMBL25079859 0.77 CCR6 (0.46) CDK2
SCHEMBL25079792 0.77 CCR6 (0.47) CDK2KDRMET
SCHEMBL25079539 0.76 CCR6 (0.47) CDK2
SCHEMBL25079808 0.76 CCR6 (0.47) CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023023534-A2 ARYL SULFONYL COMPOUNDS AS CCR6 INHIBITORS CHEMOCENTRYX, INC. (US) 2023-02-23 WO disclosed