Benzocaine

Benzocaine

SCHEMBL25100

CCOC(=O)c1ccc(N)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
CYP1A2 P05177 3/20 1.00
CYP3A4 P08684 3/20 1.00
MAOA P21397 2/20 1.00
CA1 P00915 3/20 0.68
CA2 P00918 3/20 0.68
CA12 O43570 2/20 0.68
CA7 P43166 2/20 0.68
CA9 Q16790 2/20 0.68
CA14 Q9ULX7 2/20 0.68
ESR1 P03372 1/20 0.68
ESR2 Q92731 1/20 0.68
TSHR P16473 2/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
PDE4D Q08499 1/20 0.68
NPC1 O15118 2/20 0.64
RAB9A P51151 2/20 0.64
ALDH1A1 P00352 2/20 0.64
MAPT P10636 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzocaine SCHEMBL1235972 1.00 LMNA (1.00) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL11021778 0.98 LMNA (0.96) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL944986 0.98 LMNA (0.96) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL27914401 0.98 LMNA (0.96) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL19031788 0.98 LMNA (0.96) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL15200678 0.98 LMNA (0.96) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL29029466 0.96 LMNA (0.92) LMNACYP1A2CYP3A4MAOACA1
Benzocaine SCHEMBL2389408 0.96 LMNA (0.92) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL6323309 0.94 LMNA (0.89) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL11374568 0.94 LMNA (0.89) LMNACYP1A2CYP3A4MAOACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 48198 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144801-A1 COMPOSITIONS AND METHODS FOR PREVENTING OR TREATING MUSCLE CONDITIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-28 US claimed
US-20260137637-A1 ANESTHETIC AGENT MICRO AND NANO PARTICLES, AND METHODS OF MAKING AND USING THE SAME HAAS ERIC (US) 2026-05-21 US claimed
CN-122031290-A Percutaneous permeation promoting system and preparation method and application thereof 北京工商大学 2026-05-15 CN claimed
US-12622873-B2 Composition of matter comprising liposomes embedded in a polymeric matrix and methods of using same YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2026-05-12 US claimed
EP-4110293-B1 EUTECTIC BASED ANESTHETIC COMPOSITIONS AND APPLICATIONS THEREOF UNIV NORTH CAROLINA CHAPEL HILL (US) 2026-05-06 EP claimed
EP-4735042-A1 MERCERIZED DECELLULARIZED PARTICLES FOR SLOW RELEASE APPLICATIONS AND METHODS THEREOF Spiderwort Biotechnologies Inc. (CA) 2026-05-06 EP claimed
EP-4734958-A1 TOPICAL COMPOSITION FOR PAIN RELIEF Kenvue Brands LLC (US) 2026-05-06 EP claimed
US-20260115156-A1 INJECTABLE COMPOSITION INCLUDING HYDROGEL CONTAINING ANESTHETIC AGENT UNIV KOREA RES & BUS FOUND (KR) 2026-04-30 US claimed
US-20260107921-A1 STYPTIC APPARATUS FOR PET'S CLAW OR BEAK AND METHOD FOR MANUFACTURING THE SAME OH MINHA (US) 2026-04-23 US claimed
EP-3723819-B1 WOUND DRESSING ANIMAL ETHICS PTY LTD (AU) 2026-04-22 EP claimed
EP-0002522-A1 Process for polymerizing butene-1 PHILLIPS PETROLEUM COMPANY (US) 1979-06-27 EP claimed
EP-0002521-A1 Titanium-magnesium/manganese-aluminum catalyst and process for olefin polymerization PHILLIPS PETROLEUM COMPANY (US) 1979-06-27 EP claimed
US-4148917-A PENETRATION THE PROCTER & GAMBLE COMPANY (US) 1979-04-10 US claimed
US-4147770-A ETHANOL, SALICYLIC ACID, BENZOCAINE AND VANILLIN SCHOLL, INC. (US) 1979-04-03 US claimed
US-4125730-A Preparation of -aminoalkanoic acid arylamides BANYU PHARMACEUTICAL CO., LTD. (JP) 1978-11-14 US claimed
US-4118480-A PHENOL, MENTHOL, BISMUTH SUBNITRATE, DIBUCAINE, AND PULVERIZED STARCH Stoelker, Charles V. (US) 1978-10-03 US claimed
US-4091090-A PENETRANT ACCELERATOR COMPRISING CYCLOHEXYL-SUBSTITUTED ALKANOLS JOHNSON & JOHNSON (US) 1978-05-23 US claimed
US-4083965-A ARROWROOT, CALCIUM PHOSPHATE BLUHM HENRY P 1978-04-11 US claimed
US-4064129-A Process for making quinacridone and its derivatives HARMON COLORS CORPORATION (US) 1977-12-20 US claimed
US-4041174-A INJECTING AN ESTER LOCAL ANESTHETIC ROM-AMER PHARMACEUTICALS, LTD. (US) 1977-08-09 US claimed