SCHEMBL25100560

SCHEMBL25100560

COc1cc(-c2ccc(C)cn2)ccc1-c1ccccc1-c1cc(CCc2ccc(-c3ccccn3)cc2)cc(CCc2ccc(-c3ccccn3)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.36
HCRTR2 O43614 4/20 0.36
BRS3 P32247 3/20 0.36
NR1I2 O75469 1/20 0.36
NMBR P28336 1/20 0.36
GRPR P30550 1/20 0.36
KCNH2 Q12809 1/20 0.36
SYK P43405 2/20 0.36
ERN1 O75460 1/20 0.35
WNT3A P56704 1/20 0.35
GUSB P08236 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
TGFBR1 P36897 1/20 0.34
FFAR1 O14842 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100917 0.95 CYP11B1 (0.36) BRS3MAPTMEN1KMT2AGAA
SCHEMBL21290345 0.92 HCRTR1 (0.41) HCRTR1HCRTR2BRS3NR1I2NMBR
SCHEMBL21289785 0.89 HCRTR1 (0.39) HCRTR1HCRTR2BRS3NR1I2NMBR
SCHEMBL23956228 0.89 SYK (0.40) SYKERN1GUSBALDH1A1MAPT
SCHEMBL25100909 0.88 BRS3 (0.37) HCRTR1HCRTR2BRS3NR1I2NMBR
SCHEMBL25100939 0.87 WNT3A (0.39) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100830 0.86 CYP11B1 (0.38) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100802 0.85 BRS3 (0.35) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100922 0.85 ABL1 (0.36) HCRTR1HCRTR2BRS3SYKALDH1A1
SCHEMBL25100778 0.85 NPC1 (0.50) HCRTR1HCRTR2ERN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed