SCHEMBL25100830

SCHEMBL25100830

Cc1ccc(-c2ccc(-c3ccccc3-c3cc(CCc4ccc(-c5ccccn5)cc4)cc(CCc4ccc(-c5ccccn5)cc4)c3)c(-c3ccc(-c4ccccc4)cc3)c2)nc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.38
CYP11B2 P19099 4/20 0.38
CYP3A4 P08684 2/20 0.38
BRS3 P32247 4/20 0.37
FFAR1 O14842 1/20 0.37
NR1I2 O75469 1/20 0.37
NMBR P28336 1/20 0.37
GRPR P30550 1/20 0.37
KCNH2 Q12809 1/20 0.37
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36
CYP2A6 P11509 1/20 0.36
WNT3A P56704 1/20 0.36
TGFBR1 P36897 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100976 0.95 CYP11B1 (0.42) CYP11B1CYP11B2CYP3A4BRS3FAAH
SCHEMBL26550035 0.91 TGFBR1 (0.39) CYP11B1CYP11B2BRS3FFAR1NR1I2
SCHEMBL21290071 0.90 FFAR1 (0.43) CYP11B1CYP11B2BRS3FFAR1NR1I2
SCHEMBL21290404 0.90 FFAR1 (0.43) CYP11B1CYP11B2BRS3FFAR1NR1I2
SCHEMBL26550009 0.89 TGFBR1 (0.39) CYP11B1CYP11B2BRS3FFAR1NR1I2
SCHEMBL23956272 0.89 CYP3A4 (0.43) CYP11B1CYP11B2CYP3A4CYP2A6TGFBR1
SCHEMBL26550027 0.89 FFAR1 (0.44) BRS3FFAR1NR1I2NMBRGRPR
SCHEMBL26550067 0.89 GRM5 (0.38) CYP11B1BRS3NR1I2NMBRGRPR
SCHEMBL25100939 0.89 WNT3A (0.39) CYP11B1CYP11B2CYP3A4BRS3FFAR1
SCHEMBL25100532 0.88 CYP11B1 (0.42) CYP11B1CYP11B2CYP3A4BRS3FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed