SCHEMBL25100561

SCHEMBL25100561

O=S(=O)(Oc1cccc(-c2cc(-c3ccccc3)c(-c3ccccc3-c3cc(CCc4ccc(-c5ccccc5)nc4)cc(CCc4ccc(-c5ccccc5)nc4)c3)cn2)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 3/20 0.39
CYP11B1 P15538 9/20 0.36
CYP11B2 P19099 9/20 0.36
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 2/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33
FGFR3 P22607 1/20 0.32
KDR P35968 1/20 0.32
SDHB P21912 1/20 0.32
DYRK1A Q13627 1/20 0.32
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100894 0.92 CHRM5 (0.40) CHRM5CYP11B1CYP11B2DRD2DRD1
SCHEMBL25100796 0.87 CHRM5 (0.39) CHRM5CYP11B1CYP11B2CYP3A4
SCHEMBL23956293 0.86 DYRK1A (0.36) CHRM5CYP11B1CYP11B2NR1H2NR1H3
SCHEMBL23956347 0.86 DYRK1A (0.36) CHRM5CYP11B1CYP11B2NR1H2NR1H3
SCHEMBL25100911 0.86 CHRM5 (0.35) CHRM5CYP11B1CYP11B2NR1H2NR1H3
SCHEMBL25100950 0.86 CHRM5 (0.36) CHRM5CYP11B1CYP11B2FGFR3KDR
SCHEMBL21290392 0.84 CYP11B1 (0.47) CYP11B1CYP11B2DYRK1ACYP3A4
SCHEMBL25100932 0.83 CYP11B1 (0.47) CYP11B1CYP11B2CYP3A4
SCHEMBL21290201 0.81 CYP11B1 (0.44) CYP11B1CYP11B2CYP3A4
SCHEMBL21290350 0.81 CYP11B1 (0.44) CYP11B1CYP11B2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed