SCHEMBL23956293

SCHEMBL23956293

O=S(=O)(Oc1cccc(-c2cc(-c3ccccc3)c(-c3ccccc3-c3cc(-c4ccccc4-c4ccc(-c5ccccc5)nc4)cc(-c4ccccc4-c4ccc(-c5ccccc5)nc4)c3)cn2)c1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.36
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ALOX5AP P20292 3/20 0.34
FEN1 P39748 3/20 0.34
SDHB P21912 1/20 0.34
CHRM5 P08912 1/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
DGAT1 O75907 2/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 2/20 0.33
HPGDS O60760 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
LDHA P00338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23956347 1.00 DYRK1A (0.36) DYRK1AHSD17B1HSD17B2CYP11B1CYP11B2
SCHEMBL23956362 0.94 DYRK1A (0.40) DYRK1AHSD17B1HSD17B2CYP11B1CYP11B2
SCHEMBL23956219 0.91 LDHA (0.40) DYRK1AALOX5APFEN1SDHBDGAT1
SCHEMBL24291876 0.87 ADORA2A (0.39) DYRK1AALOX5APFEN1CHRM5ADORA2A
SCHEMBL24291878 0.87 ADORA2A (0.39) DYRK1AALOX5APFEN1CHRM5ADORA2A
SCHEMBL25100561 0.86 CHRM5 (0.39) DYRK1ACYP11B1CYP11B2SDHBCHRM5
SCHEMBL22175451 0.86 PDK2 (0.37) CHRM5ADORA2AADORA1
SCHEMBL23956295 0.85 HSD17B1 (0.37) HSD17B1HSD17B2ALOX5APFEN1CHRM5
SCHEMBL23956284 0.85 ALOX5AP (0.36) CYP11B1CYP11B2ALOX5APFEN1CHRM5
SCHEMBL22175327 0.84 LDHA (0.41) DYRK1AALOX5APFEN1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed