SCHEMBL25100950

SCHEMBL25100950

O=S(=O)(Oc1cc(-c2cccc(-c3ccccc3)c2)ncc1-c1ccccc1-c1cc(CCc2ccc(-c3ccccc3)nc2)cc(CCc2ccc(-c3ccccc3)nc2)c1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.36
CYP11B1 P15538 10/20 0.36
CYP11B2 P19099 10/20 0.36
WNT3A P56704 2/20 0.32
CYP3A4 P08684 1/20 0.31
FGFR3 P22607 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100796 0.95 CHRM5 (0.39) CHRM5CYP11B1CYP11B2CYP3A4
SCHEMBL23956295 0.88 HSD17B1 (0.37) CHRM5
SCHEMBL25100561 0.86 CHRM5 (0.39) CHRM5CYP11B1CYP11B2CYP3A4FGFR3
SCHEMBL25100806 0.84 USP1 (0.38)
SCHEMBL21289938 0.84 CYP11B1 (0.42) CYP11B1CYP11B2WNT3ACYP3A4
SCHEMBL23956284 0.83 ALOX5AP (0.36) CHRM5CYP11B1CYP11B2
SCHEMBL25100894 0.83 CHRM5 (0.40) CHRM5CYP11B1CYP11B2WNT3A
SCHEMBL25100508 0.83 LDHA (0.34) CHRM5
SCHEMBL25100764 0.82 CHRM5 (0.36) CHRM5CYP11B1CYP11B2WNT3ACYP3A4
SCHEMBL21290201 0.80 CYP11B1 (0.44) CYP11B1CYP11B2WNT3ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed