SCHEMBL2510429

SCHEMBL2510429

Cc1nccn1-c1ccc(NN2C=C(N3c4ccccc4CC3CO)C3=C(CNC(C)C3)C2)cc1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
PORCN Q9H237 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2509408 0.79 ADH5 (0.34) CYP3A4CYP2D6PORCN
SCHEMBL2483928 0.67 SYK (0.32) CYP3A4CYP2D6PORCN
SCHEMBL2483931 0.67 SYK (0.32) CYP3A4CYP2D6PORCN
SCHEMBL2498451 0.66 PDE3B (0.36) CYP3A4CYP2D6PORCN
SCHEMBL2477814 0.66 ROCK2 (0.39) CYP3A4CYP2D6PORCN
SCHEMBL2446909 0.66 ROCK2 (0.39) CYP3A4CYP2D6PORCN
SCHEMBL2477810 0.66 ROCK2 (0.39) CYP3A4CYP2D6PORCN
SCHEMBL2843972 0.62 ROCK2 (0.33)
SCHEMBL2449527 0.62 ROCK2 (0.33)
SCHEMBL2848556 0.61 MAPT (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367826-A1 MODULATORS OF AMYLOID BETA. AstraZeneca AB (SE) 2011-09-28 EP disclosed
WO-2010053438-A1 MODULATORS OF AMYLOID BETA. ASTRAZENECA AB (SE) 2010-05-14 WO disclosed