SCHEMBL2512431

SCHEMBL2512431

CC(C)OC(=O)[C@H](C)NP(=O)(Oc1ccccc1)Oc1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTN3A1 O00481 12/20 0.50
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2521572 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL16690101 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL2521573 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL2549985 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL30208193 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL16081101 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL2510991 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL850195 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL2510990 1.00 BTN3A1 (0.50) BTN3A1CYP3A4CYP2C9MEN1KMT2A
SCHEMBL19821287 0.95 BTN3A1 (0.47) BTN3A1CYP3A4CYP2C9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 267 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016181313-A1 A PROCESS FOR THE PREPARATION OF SOFOSBUVIR INTERMEDIATES & ITS POLYMORPH LUPIN LIMITED (IN) 2016-11-17 WO claimed
EP-2552930-A2 NUCLEOSIDE PHOSPHORAMIDATES Gilead Pharmasset LLC (US) 2013-02-06 EP claimed
WO-2011123645-A2 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2011-10-06 WO claimed
EP-4705313-A2 4'-SUBSTITUTED NUCLEOSIDES AND NUCLEOTIDES AS ANTIVIRAL AGENTS The Scripps Research Institute (US) 2026-03-11 EP disclosed
US-20260062437-A1 ANTIVIRAL COMPOUNDS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2026-03-05 US disclosed
WO-2025235664-A1 PURINE NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2025-11-13 WO disclosed
US-20250282803-A1 DIDEHYDRO-3'-DEOXY-4'-ETHYNYLTHYMIDINES AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS ROME THERAPEUTICS, INC. 2025-09-11 US disclosed
US-20250109163-A1 NUCLEOTIDE HEMI-SULFATE SALT FOR THE TREATMENT OF HEPATITIS C VIRUS Atea Pharmaceuticals, Inc. (US) 2025-04-03 US disclosed
WO-2025049569-A2 EXTENDED PURINE TRICYCLIC AND BICYCLIC NUCLEOSIDES AND NUCLEOTIDES FOR USE AS ANTIVIRAL THERAPEUTICS UNIVERSITY OF MARYLAND, BALTIMORE COUNTY (US) 2025-03-06 WO disclosed
EP-4511381-A1 DIDEHYDRO-3'-DEOXY-4'-ETHYNYLTHYMIDINES AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS Rome Therapeutics, Inc. (US) 2025-02-26 EP disclosed
US-20250057867-A1 NUCLEOSIDE PHOSPHORAMIDATES GILEAD SCIENCES INC (US) 2025-02-20 US disclosed
US-20110251152-A1 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2011-10-13 US disclosed
WO-2011123668-A2 STEREOSELECTIVE SYNTHESIS OF PHOSPHORUS CONTAINING ACTIVES PHARMASSET, INC. (US) 2011-10-06 WO disclosed
WO-2011123645-A2 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2011-10-06 WO disclosed
WO-2011123672-A1 PURINE NUCLEOSIDE PHOSPHORAMIDATE PHARMASSET, INC. (US) 2011-10-06 WO disclosed
WO-2011123645-A2 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2011-10-06 WO disclosed
US-20110245484-A1 STEREOSELECTIVE SYNTHESIS OF PHOSPHORUS CONTAINING ACTIVES PHARMASSET, INC. (US) 2011-10-06 US disclosed
WO-2010135569-A1 N- [ (2 ' R) -2 ' -DEOXY-2 ' -FLUORO-2 ' -METHYL-P-PHENYL-5 ' -URIDYLYL] -L-ALANINE 1-METHYLETHYL ESTER AND PROCESS FOR ITS PRODUCTION PHARMASSET, INC. (US) 2010-11-25 WO disclosed
US-20100298257-A1 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2010-11-25 US disclosed
US-20100298257-A1 NUCLEOSIDE PHOSPHORAMIDATES PHARMASSET, INC. (US) 2010-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260062437-A1 ANTIVIRAL COMPOUNDS ZC3HAV1, IFNAR1, IRF3 BTN3A1 3335/4885CYP3A4 2578/4885CYP2C9 3181/4885
US-20250109163-A1 NUCLEOTIDE HEMI-SULFATE SALT FOR THE TREATMENT OF HEPATITIS C VIRUS HAVCR2, HCCS, SLC10A1 BTN3A1 3397/4885CYP3A4 1930/4885CYP2C9 2514/4885
US-20250057867-A1 NUCLEOSIDE PHOSPHORAMIDATES PNP, RNGTT, NSUN2 BTN3A1 3601/4885CYP3A4 3916/4885CYP2C9 4098/4885
US-20100298257-A1 NUCLEOSIDE PHOSPHORAMIDATES PNP, RNGTT, NSUN2 BTN3A1 3738/4885CYP3A4 3811/4885CYP2C9 3971/4885
US-20110245484-A1 STEREOSELECTIVE SYNTHESIS OF PHOSPHORUS CONTAINING ACTIVES PPA1, ENPP1, ITPA BTN3A1 3359/4885CYP3A4 1919/4885CYP2C9 1843/4885
US-20250282803-A1 DIDEHYDRO-3'-DEOXY-4'-ETHYNYLTHYMIDINES AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS DTYMK, DCK, POLK BTN3A1 3447/4885CYP3A4 596/4885CYP2C9 932/4885
US-20110251152-A1 NUCLEOSIDE PHOSPHORAMIDATES PNP, RNGTT, NSUN2 BTN3A1 3601/4885CYP3A4 3916/4885CYP2C9 4098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.