SCHEMBL25130366

SCHEMBL25130366

COc1c(Br)cc2c(Cl)ccnc2c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
HSP90AA1 P07900 3/20 0.36
HSP90AB1 P08238 1/20 0.36
NQO2 P16083 1/20 0.35
AXL P30530 1/20 0.33
PRKCI P41743 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CHUK O15111 1/20 0.32
NSD2 O96028 1/20 0.32
CASP6 P55212 1/20 0.32
G6PD P11413 1/20 0.32
BRAF P15056 1/20 0.31
PIK3CA P42336 1/20 0.31
DYRK1A Q13627 1/20 0.31
KDM4E B2RXH2 3/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
TDP1 Q9NUW8 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29923920 0.75 HSP90AA1 (0.50) HSP90AA1HSP90AB1NSD2CASP6G6PD
SCHEMBL27163581 0.74 KDM4E (0.35) HSP90AA1HSP90AB1AXLPRKCIKDM4E
SCHEMBL3305107 0.73 NQO2 (0.39) ALOX5APFEN1NQO2CA2CA4
SCHEMBL22233797 0.73 KDM4E (0.39) HSP90AA1AXLPRKCIKDM4EMEN1
SCHEMBL24010300 0.72 KDM4E (0.40) HSP90AA1G6PDDYRK1AKDM4EMEN1
SCHEMBL6599333 0.72 NQO2 (0.38) NQO2CA2CA4NSD2CASP6
SCHEMBL24009363 0.71 PDE2A (0.42) HSP90AA1HSP90AB1G6PDDYRK1AKDM4E
SCHEMBL1878775 0.71 KDM4E (0.37) HSP90AA1HSP90AB1AXLPRKCIKDM4E
SCHEMBL25130340 0.70 MAPT (0.51) KDM4EALDH1A1TP53LMNAMAPT
SCHEMBL30666114 0.70 HSP90AA1 (0.38) HSP90AA1HSP90AB1AXLPRKCIG6PD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023051628-A1 SOS1 INHIBITORS HAVING PYRIDO SIX-MEMBERED RING STRUCTURE 上海海和药物研究开发股份有限公司 2023-04-06 WO disclosed