SCHEMBL29923920

SCHEMBL29923920

COc1cc(Br)c2nccc(Cl)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.50
HSP90AB1 P08238 1/20 0.50
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
KDM4E B2RXH2 3/20 0.38
POLB P06746 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
DYRK1A Q13627 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP4B1 P13584 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9073416 0.83 HSP90AA1 (0.50) HSP90AA1HSP90AB1CCR1CCR5CCR8
SCHEMBL2270856 0.82 HSP90AA1 (0.52) HSP90AA1HSP90AB1CCR1CCR5CCR8
SCHEMBL24916289 0.81 NSD2 (0.50) CCR1CCR5CCR8KDM4ENOS3
SCHEMBL24916103 0.80 NOS3 (0.41) HSP90AA1CCR1CCR5CCR8KDM4E
SCHEMBL29923344 0.80 CCR1 (0.39) HSP90AA1HSP90AB1CCR1CCR5CCR8
SCHEMBL29924149 0.80 NOS3 (0.41) HSP90AA1CCR1CCR5CCR8KDM4E
SCHEMBL31392519 0.79 KDM4E (0.39) HSP90AA1HSP90AB1CCR1CCR5CCR8
SCHEMBL25130366 0.75 ALOX5AP (0.39) HSP90AA1HSP90AB1KDM4EDYRK1ACYP3A4
SCHEMBL31728793 0.75 KDM4E (0.49) KDM4EPOLBCYP1A1CYP1B1KMT2A
SCHEMBL5262975 0.73 PDGFRB (0.42) CCR1CCR5CCR8KDM4ENOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed