SCHEMBL25135

SCHEMBL25135

O=C(Oc1cccc2ccccc12)c1ccccc1O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.77
GAA P10253 3/20 0.77
POLB P06746 1/20 0.77
HSD17B10 Q99714 5/20 0.63
ALDH1A1 P00352 3/20 0.63
HPGD P15428 2/20 0.63
KDM4E B2RXH2 1/20 0.63
ESR1 P03372 5/20 0.61
ESR2 Q92731 5/20 0.61
MEN1 O00255 3/20 0.61
MAPT P10636 3/20 0.56
HTT P42858 1/20 0.56
ALOX15 P16050 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
JAK2 O60674 1/20 0.55
USP2 O75604 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
EGFR P00533 1/20 0.54
PGR P06401 1/20 0.53
PTGS1 P23219 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392731 1.00 KMT2A (0.77) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL3757751 0.90 KMT2A (0.70) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL30185780 0.89 HSD17B10 (0.67) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL8367791 0.88 KMT2A (0.78) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL27773732 0.87 KMT2A (1.00) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL11754236 0.86 KMT2A (0.76) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL11358096 0.83 KMT2A (0.62) KMT2AGAAPOLBHSD17B10ALDH1A1
Acetic Acid SCHEMBL27380873 0.83 KMT2A (0.62) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL10686808 0.82 HSD17B10 (0.71) KMT2AGAAPOLBHSD17B10ALDH1A1
SCHEMBL3635482 0.82 HPGD (0.76) KMT2AGAAPOLBHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2230 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
US-11648198-B2 Expandable gastroretentive dosage form CLEXIO BIOSCIENCES LTD. (IL) 2023-05-16 US claimed
CN-115607556-A Medicine for preventing and treating asthma, chronic obstructive pulmonary disease, allergic diseases, etc 刘力 2023-01-17 CN claimed
CN-115607516-A Medicine for preventing and treating cold or viral diseases 刘力 2023-01-17 CN claimed
WO-2021054927-A2 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2021-03-25 WO claimed
EP-3263145-B1 ANTIMICROBIAL COMPOSITIONS AND METHODS FOR LOCKING CATHETERS BECTON DICKINSON CO (US) 2021-01-20 EP claimed
US-20200405635-A1 EXPANDABLE GASTRORETENTIVE DOSAGE FORM CLEXIO BIOSCIENCES LTD. (IL) 2020-12-31 US claimed
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2020-02-13 US claimed
EP-2822532-B1 AQUEOUS POLYURETHANE DISPERSION IN THE TREATMENT OF ACNE COVESTRO DEUTSCHLAND AG (DE) 2018-09-19 EP claimed
US-9872941-B2 Antimicrobial compositions and methods for locking catheters BECTON, DICKINSON AND COMPANY (US) 2018-01-23 US claimed
WO-1998020864-A9 USE OF SELECTED NON-STEROIDAL ANTIINFLAMMATORY COMPOUNDS FOR THE PREVENTION AND THE TREATMENT OF NEURODEGENERATIVE DISEASES 1998-08-27 WO claimed
WO-1998020864-A2 USE OF SELECTED NON-STEROIDAL ANTIINFLAMMATORY COMPOUNDS FOR THE PREVENTION AND THE TREATMENT OF NEURODEGENERATIVE DISEASES UNIVERSITA' DEGLI STUDI DI BRESCIA - DIPARTIMENTO DI SCIENZE BIOMEDICHE (IT) 1998-05-22 WO claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
US-5536419-A Procedure for extraction of polyhydroxyalkanoates from halophilic bacteria which contain them REPSOL QUIMICA S.A. (ES) 1996-07-16 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
EP-0622462-A1 Procedure for the extraction of polyhydroxyalkanoates from halophilic bacteria which contain them REPSOL QUIMICA S.A. (ES) 1994-11-02 EP claimed
US-4432966-A SUSTAINED RELEASE ROUSSEL-UCLAF (FR) 1984-02-21 US claimed