SCHEMBL25147754

SCHEMBL25147754

Cc1cc(C#N)nnc1N1CCc2ncc(C(C)(O)C(F)(F)F)cc2C1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.33
CYP11B1 P15538 2/20 0.33
AR P10275 1/20 0.31
KDM4E B2RXH2 1/20 0.30
PDK1 Q15118 2/20 0.30
PDK2 Q15119 2/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KDR P35968 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31660077 1.00 CYP11B2 (0.33) CYP11B2CYP11B1ARKDM4EPDK1
SCHEMBL25153188 0.89 KDM4E (0.35) KDM4EKDR
SCHEMBL30370412 0.89 KDM4E (0.35) KDM4EKDR
SCHEMBL25147763 0.85 PDK2 (0.35) CYP11B2CYP11B1ARPDK1PDK2
SCHEMBL31659690 0.85 PDK2 (0.35) CYP11B2CYP11B1ARPDK1PDK2
SCHEMBL25147750 0.85 SMO (0.34) CYP11B2CYP11B1ARHDAC6KDR
SCHEMBL31659593 0.85 SMO (0.34) CYP11B2CYP11B1ARHDAC6KDR
SCHEMBL31659721 0.81 GRIN2D (0.32) KDM4E
SCHEMBL25148366 0.81 GRIN2D (0.32) KDM4E
SCHEMBL25147753 0.80 KDM4E (0.33) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed