SCHEMBL25148403

SCHEMBL25148403

Cc1cc(C#N)cnc1N1CCc2ncc(C(F)F)cc2C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
TYK2 P29597 2/20 0.35
JAK3 P52333 2/20 0.35
P2RX3 P56373 10/20 0.34
P2RX2 Q9UBL9 10/20 0.34
PDE10A Q9Y233 1/20 0.33
KCNJ1 P48048 2/20 0.33
USP14 P54578 1/20 0.32
PLK1 P53350 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31659875 1.00 JAK2 (0.35) JAK2JAK1TYK2JAK3P2RX3
SCHEMBL31659770 0.85 JAK2 (0.37) JAK2JAK1TYK2JAK3PDE10A
SCHEMBL30331871 0.85 JAK2 (0.37) JAK2JAK1TYK2JAK3PDE10A
SCHEMBL25147771 0.85 JAK2 (0.37) JAK2JAK1TYK2JAK3PDE10A
SCHEMBL31659482 0.85 JAK2 (0.38) JAK2JAK1TYK2JAK3P2RX3
SCHEMBL25148210 0.85 JAK2 (0.38) JAK2JAK1TYK2JAK3P2RX3
SCHEMBL25148356 0.84 P2RX3 (0.32) P2RX3P2RX2PDE10APLK1
SCHEMBL31660328 0.84 P2RX3 (0.32) P2RX3P2RX2PDE10APLK1
SCHEMBL25148376 0.83 SCN10A (0.39) JAK2JAK1TYK2JAK3P2RX3
SCHEMBL30332227 0.83 SCN10A (0.39) JAK2JAK1TYK2JAK3P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed