SCHEMBL25162437

SCHEMBL25162437

C=CC(=O)Nc1cccc(C)c1Nc1cc2c(cn1)cc(-c1cc(OC)cc(OC)c1)c(=O)n2CCCN1CCOCC1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 17/20 0.72
FGFR1 P11362 9/20 0.61
FGFR2 P21802 1/20 0.61
FGFR3 P22607 1/20 0.61
BTK Q06187 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25162435 0.94 FGFR4 (0.74) FGFR4FGFR1FGFR2FGFR3
SCHEMBL25162439 0.94 FGFR4 (0.74) FGFR4FGFR1FGFR2FGFR3
SCHEMBL25162206 0.89 FGFR4 (0.80) FGFR4FGFR1FGFR2FGFR3
SCHEMBL27428516 0.88 FGFR4 (0.66) FGFR4FGFR1FGFR2FGFR3
SCHEMBL25162186 0.88 FGFR4 (0.81) FGFR4FGFR1FGFR2FGFR3
SCHEMBL28694174 0.86 FGFR4 (0.57) FGFR4FGFR1FGFR2FGFR3BTK
SCHEMBL25162205 0.86 FGFR4 (0.72) FGFR4FGFR1FGFR2FGFR3
SCHEMBL30365929 0.86 FGFR4 (0.70) FGFR4FGFR1FGFR2FGFR3BTK
SCHEMBL15434012 0.84 FGFR4 (1.00) FGFR4FGFR1FGFR2FGFR3
SCHEMBL28679307 0.83 FGFR4 (0.68) FGFR4FGFR1FGFR2FGFR3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4393921-A1 NALIDINONE COMPOUND AS FGFR4 INHIBITOR AND USE THEREOF Wenzhou Medical University (CN) 2024-07-03 EP disclosed
CN-113912602-B 2-oxo-1, 2-dihydro-1, 6-naphthyridine-7-yl compound and preparation method and application thereof 温州医科大学 2023-05-05 CN disclosed
WO-2023060904-A1 NALIDINONE COMPOUND AS FGFR4 INHIBITOR AND USE THEREOF 温州医科大学 2023-04-20 WO disclosed
CN-113912602-A 2-oxo-1, 2-dihydro-1, 6-naphthyridine-7-based compound and preparation method and application thereof 温州医科大学 2022-01-11 CN disclosed