SCHEMBL25164705

SCHEMBL25164705

CC(C)c1ncc2cnn(CC(F)F)c2n1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.38
HTR2C P28335 8/20 0.38
HTR2B P41595 4/20 0.34
USP1 O94782 3/20 0.32
HTR1A P08908 2/20 0.30
ADRA2A P08913 2/20 0.30
ADRA2B P18089 2/20 0.30
ADRA2C P18825 2/20 0.30
HTR1D P28221 1/20 0.30
HTR7 P34969 1/20 0.30
HTR4 Q13639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18898669 0.82 XDH (0.36) HTR2AHTR2CHTR2B
SCHEMBL25164185 0.81 HTR2A (0.34) HTR2AHTR2CHTR2BUSP1
SCHEMBL25164210 0.80 CYP17A1 (0.38) HTR2AHTR2CUSP1
SCHEMBL25164208 0.79 RIPK1 (0.37) HTR2AHTR2CUSP1
SCHEMBL29202302 0.78 HTR2A (0.33) HTR2AHTR2CHTR2B
SCHEMBL30328297 0.78 HTR2A (0.33) HTR2AHTR2CHTR2B
SCHEMBL25164322 0.75 PDE10A (0.33)
SCHEMBL19421539 0.73 PI4KA (0.34)
SCHEMBL17807781 0.71 AURKA (0.40)
SCHEMBL30174416 0.71 HTR2A (0.40) HTR2AHTR2CHTR2BHTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064343-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2023-04-20 WO disclosed