SCHEMBL25200397

SCHEMBL25200397

O=CNc1n[nH]c2ccc(Br)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 3/20 0.53
JAK2 O60674 3/20 0.53
FADS1 O60427 2/20 0.51
DYRK1A Q13627 6/20 0.47
CSNK2A1 P68400 2/20 0.47
PRKD3 O94806 2/20 0.47
MAP4K4 O95819 2/20 0.47
CSF1R P07333 2/20 0.47
FLT3 P36888 2/20 0.47
CLK2 P49760 2/20 0.47
MAP4K2 Q12851 2/20 0.47
NTRK3 Q16288 2/20 0.47
AURKB Q96GD4 2/20 0.47
CLK4 Q9HAZ1 2/20 0.47
CDK2 P24941 2/20 0.47
DCLK1 O15075 1/20 0.47
CHEK2 O96017 1/20 0.47
FER P16591 1/20 0.47
MARK3 P27448 1/20 0.47
FLT4 P35916 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2671952 0.78 PDPK1 (0.58) PDPK1JAK2FADS1DYRK1ACSNK2A1
SCHEMBL26393980 0.77 GSK3B (0.57) JAK2DYRK1ACDK2GSK3BAXL
SCHEMBL11748390 0.77 FADS1 (0.54) FADS1GSK3B
SCHEMBL28079288 0.77 NTRK1 (0.45) CDK2GSK3BNTRK1GSK3APRKAA1
SCHEMBL11754096 0.76 TRPA1 (0.50) PDPK1FADS1FLT3CDK2MAPK8
Hydrochloric Acid SCHEMBL8487463 0.75 TRPA1 (0.49) PDPK1FADS1FLT3CDK2MAPK8
SCHEMBL660142 0.75 PDPK1 (0.58) PDPK1JAK2FADS1DYRK1ACSNK2A1
SCHEMBL28079409 0.75 TRPA1 (0.49) PDPK1FADS1FLT3CDK2MAPK8
SCHEMBL6487193 0.73 DYRK1A (0.51) PDPK1JAK2FADS1DYRK1ACSNK2A1
SCHEMBL15484549 0.73 DYRK1A (0.51) PDPK1JAK2FADS1DYRK1ACSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078337-A1 CDK8/19 DUAL INHIBITORS AND METHODS OF USE INSILICO MEDICINE IP LIMITED (CN) 2023-05-11 WO disclosed
WO-2023078337-A1 CDK8/19 DUAL INHIBITORS AND METHODS OF USE INSILICO MEDICINE IP LIMITED (CN) 2023-05-11 WO disclosed