SCHEMBL25224263

SCHEMBL25224263

C[C@H]1CN(C(=O)O)CCCN1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC2 Q13490 1/20 0.49
CA2 P00918 1/20 0.36
CHKA P35790 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
REN P00797 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
CHRNB3 Q05901 1/20 0.31
CHRNA6 Q15825 1/20 0.31
CNR1 P21554 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033981 1.00 BIRC2 (0.49) BIRC2CA2CHKAHRH4ALDH1A1
SCHEMBL28621816 0.94 BIRC2 (0.51) BIRC2CA2CHKAHRH4ALDH1A1
SCHEMBL190023 0.88 BIRC2 (0.47) BIRC2CA2CHKAHRH4REN
SCHEMBL190024 0.88 BIRC2 (0.47) BIRC2CA2CHKAHRH4REN
SCHEMBL1181669 0.88 BIRC2 (0.47) BIRC2CA2CHKAHRH4REN
SCHEMBL15825441 0.79 REN (0.36) BIRC2CA2CHKALMNAREN
SCHEMBL20139833 0.78 BIRC2 (0.37) BIRC2ALDH1A1LMNARENMEN1
SCHEMBL24322743 0.78 BIRC2 (0.51) BIRC2CA2CHKAHRH4ALDH1A1
SCHEMBL2898103 0.75 HPGD (0.48) BIRC2ALDH1A1MEN1KMT2AMAPT
SCHEMBL31540 0.75 HPGD (0.48) BIRC2ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4441054-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER Boehringer Ingelheim International GmbH (DE) 2024-10-09 EP disclosed
WO-2023099623-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed
WO-2023099592-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed