SCHEMBL252280

SCHEMBL252280

Brc1ccccc1C1OCCO1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.46
HTR2B P41595 5/20 0.46
KDM1A O60341 3/20 0.45
HTR2A P28223 3/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 1/20 0.44
RCOR1 Q9UKL0 1/20 0.37
BRD4 O60885 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29571908 1.00 HTR2C (0.46) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL1043098 0.91 HTR2C (0.43) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL29384288 0.91 HTR2C (0.43) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL11030273 0.90 HTR2C (0.42) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL3727526 0.83 TSHR (0.36) HTR2CHTR2BHTR2ASLC6A2SLC6A4
SCHEMBL24216729 0.79 KDM1A (0.42) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL30409857 0.79 KDM1A (0.42) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL29946544 0.79 NSD2 (0.36) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL11632118 0.79 HTR2C (0.41) HTR2CHTR2BKDM1AHTR2ASLC6A2
SCHEMBL26132936 0.79 KDM1A (0.34) HTR2CHTR2BKDM1AHTR2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 195 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102603797-A Phosphine imide ligand (E)-(2-(diphenyl phosphino) benzylidene) hydrazine as well as synthetic method and application of phosphine imide ligand (E)-(2-(diphenyl phosphino) benzylidene) hydrazine UNIV NANKAI 2012-07-25 CN claimed
EP-4618974-A1 OREXIN RECEPTOR AGONISTS Merck Sharp & Dohme LLC (US) 2025-09-24 EP disclosed
US-20240277848-A1 SURFACE-MODIFIED NANOPARTICLE KYOTO UNIVERSITY (JP) 2024-08-22 US disclosed
WO-2024107615-A1 OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME LLC (US) 2024-05-23 WO disclosed
WO-2024107615-A1 OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME LLC (US) 2024-05-23 WO disclosed
EP-4353680-A1 SURFACE-MODIFIED NANOPARTICLE Kyoto University (JP) 2024-04-17 EP disclosed
CN-117460698-A Surface-modified nanoparticles 国立大学法人京都大学 2024-01-26 CN disclosed
US-20240018161-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2024-01-18 US disclosed
US-20240018161-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2024-01-18 US disclosed
US-20240018161-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2024-01-18 US disclosed
EP-0391451-A1 Fungicides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-10-10 EP disclosed
EP-0387923-A2 Fungicides ZENECA LIMITED (GB) 1990-09-19 EP disclosed
US-4892885-A CARDIOTONICS, DIURETICS AMERICAN CYANAMID COMPANY 1990-01-09 US disclosed
US-4877801-A 1-Aryl-1-(1H-azol-1-ylalkyl)-1,3-dihydroisobenzofurans, related derivatives and pharmaceutical compositions thereof useful as antifungals SCHERING CORPORATION (US) 1989-10-31 US disclosed
CN-1032782-A Bactericide ICI PLC (GB) 1989-05-10 CN disclosed
EP-0307103-A2 Fungicides ZENECA LIMITED (GB) 1989-03-15 EP disclosed
US-4737508-A 1-aryl-1-(1H-azol-1-ylalkyl)-1,3-dihydroisobenzofurans, related derivatives and pharmaceutical compositions thereof useful as antifungals SCHERING CORPORATION (US) 1988-04-12 US disclosed
CN-87103623-A Fungicidal agents ICI PLC (GB) 1988-02-24 CN disclosed
EP-0242081-A1 Fungicides ZENECA LIMITED (GB) 1987-10-21 EP disclosed
US-4532237-A Treating cardiovascular disorders MERCK & CO., INC. (US) 1985-07-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018161-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1G, SCNN1B HTR2C 4306/4885HTR2B 4262/4885KDM1A 4670/4885
US-20240277848-A1 SURFACE-MODIFIED NANOPARTICLE EPCAM, CD63, CD22 HTR2C 3462/4885HTR2B 1694/4885KDM1A 2123/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.