SCHEMBL25233154

SCHEMBL25233154

Clc1cc2nccn2cc1Br

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.41
MAOB P27338 1/20 0.38
TGFBR1 P36897 9/20 0.37
KEAP1 Q14145 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
JAK2 O60674 1/20 0.32
RET P07949 1/20 0.32
AKT1 P31749 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
AXL P30530 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23302224 0.85 MAOB (0.38) DYRK1AMAOBTGFBR1KEAP1L3MBTL1
SCHEMBL22490652 0.82 MAOB (0.43) DYRK1AMAOBTGFBR1KEAP1L3MBTL1
SCHEMBL24087290 0.77 TGFBR1 (0.46) DYRK1AMAOBTGFBR1KEAP1MEN1
SCHEMBL22715717 0.77 MAOB (0.40) DYRK1AMAOBTGFBR1KEAP1L3MBTL1
SCHEMBL24087352 0.77 TGFBR1 (0.38) DYRK1ATGFBR1KEAP1L3MBTL1MEN1
SCHEMBL407441 0.77 L3MBTL1 (0.49) DYRK1ATGFBR1KEAP1L3MBTL1MEN1
SCHEMBL1911469 0.77 DYRK1A (0.38) DYRK1ATGFBR1KEAP1L3MBTL1MEN1
Bromide SCHEMBL29677074 0.76 MAOB (0.40) DYRK1AMAOBTGFBR1KEAP1MEN1
Hydrochloric Acid SCHEMBL31647268 0.76 L3MBTL1 (0.47) DYRK1ATGFBR1KEAP1L3MBTL1MEN1
SCHEMBL21246775 0.74 DYRK1A (0.45) DYRK1AMAOBTGFBR1KEAP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090330-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2026-04-30 WO disclosed
WO-2024220891-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2024-10-24 WO disclosed
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2023-09-28 US disclosed
US-20230183237-A1 COMPETITIVE AND NONCOMPETITIVE INHIBITORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M5 VANDERBILT UNIVERSITY 2023-06-15 US disclosed
US-20230183237-A1 COMPETITIVE AND NONCOMPETITIVE INHIBITORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M5 VANDERBILT UNIVERSITY 2023-06-15 US disclosed
US-20230183237-A1 COMPETITIVE AND NONCOMPETITIVE INHIBITORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M5 VANDERBILT UNIVERSITY 2023-06-15 US disclosed
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303569-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS C3AR1, C9, C1R DYRK1A 4426/4885MAOB 503/4885TGFBR1 2049/4885
US-20230183237-A1 COMPETITIVE AND NONCOMPETITIVE INHIBITORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M5 CHRM5, CHRM1, CHRM2 DYRK1A 1086/4885MAOB 168/4885TGFBR1 260/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.