SCHEMBL25237476

SCHEMBL25237476

CC(=O)c1ccnc(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.60
DDB1 Q16531 1/20 0.54
CRBN Q96SW2 1/20 0.54
GPR119 Q8TDV5 9/20 0.54
CHRNA7 P36544 1/20 0.53
MAPT P10636 2/20 0.51
PTPN11 Q06124 1/20 0.50
CKS1B P61024 1/20 0.48
SKP1 P63208 1/20 0.48
SKP2 Q13309 1/20 0.48
MAP4K4 O95819 1/20 0.47
POLB P06746 1/20 0.46
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29319392 0.90 ACHE (0.60) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL7136906 0.90 ACHE (0.63) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL27213788 0.88 ACHE (0.61) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL30995427 0.88 ACHE (0.61) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL31706344 0.88 ACHE (0.61) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL29319390 0.87 ACHE (0.57) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL7161944 0.85 ACHE (0.58) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL15286547 0.85 ACHE (0.62) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL19015403 0.84 ACHE (0.61) ACHEDDB1CRBNGPR119CHRNA7
SCHEMBL30166226 0.84 ACHE (0.61) ACHEDDB1CRBNGPR119CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023110843-A1 HETEROBICYCLIC DERIVATIVES AS ITK INHIBITORS ALMIRALL, S.A. (ES) 2023-06-22 WO disclosed