SCHEMBL25245166

SCHEMBL25245166

CC(C)(Cc1ccc(Br)cc1)S(N)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 8/20 0.44
CA1 P00915 6/20 0.44
CA9 Q16790 6/20 0.44
CA5A P35218 1/20 0.44
CA12 O43570 4/20 0.40
CA7 P43166 1/20 0.40
CA4 P22748 1/20 0.38
PTGES2 Q9H7Z7 2/20 0.38
HTR2A P28223 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
PLCG1 P19174 1/20 0.36
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9131072 0.82 CA2 (0.53) CA2HTR2ATAAR1
SCHEMBL5145167 0.80 SLC6A2 (0.54) CA2CA1CA9CA5ACA12
SCHEMBL9085340 0.79 CA2 (0.56) CA2CA1CA9CA5ACA12
SCHEMBL28458665 0.78 CA1 (0.54) CA2CA1CA9CA5ACA12
SCHEMBL21448664 0.77 CA2 (0.38) CA2CA1CA9CA5ACA12
SCHEMBL256214 0.73 SLC6A2 (0.61) HTR2ATAAR1IDO1
SCHEMBL1737226 0.73 ESR1 (0.43) HTR2ATAAR1IDO1
SCHEMBL799906 0.72 ESR1 (0.58) HTR2ATAAR1IDO1
SCHEMBL30338274 0.72 TAAR1 (0.43) HTR2ATAAR1IDO1
SCHEMBL751764 0.71 PLCG1 (0.41) CA2CA1CA9CA5ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109912-A1 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF BEIGENE, LTD. (KY) 2023-06-22 WO disclosed