SCHEMBL25246721

SCHEMBL25246721

N[C@@H](COC(=O)C(F)(F)F)Cc1c(Cl)ccnc1F

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP3A4 P08684 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
DPP4 P27487 1/20 0.30
DPP9 Q86TI2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL30490495 0.76 SLC6A2 (0.34) KDM4EALDH1A1POLBDPP4DPP9
SCHEMBL25789569 0.70 PNMT (0.40)
SCHEMBL4358436 0.68 DPP4 (0.37) DPP4
SCHEMBL588955 0.68 DPP4 (0.43) DPP4
SCHEMBL22863924 0.66 CFTR (0.32) GAAAAK1
SCHEMBL25191542 0.64 GAA (0.40) GAAKMT2ATDP1
SCHEMBL25199133 0.64 LOXL2 (0.39) GAAKDM4EKMT2ATDP1DPP4
SCHEMBL29009936 0.63 FFAR1 (0.43)
Hydrochloric Acid SCHEMBL25196993 0.62 LOXL2 (0.38) GAAKDM4EALDH1A1KMT2ATDP1
SCHEMBL13729617 0.62 DPP4 (0.37) CYP3A4DPP4DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4456892-A1 BICYCLIC INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE, COMPOSITIONS AND USES THEREOF President and Fellows of Harvard College (US) 2024-11-06 EP disclosed
WO-2023129512-A1 BICYCLIC INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE, COMPOSITIONS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-07-06 WO disclosed