SCHEMBL25249404

SCHEMBL25249404

O=C(O)c1cc(Br)n2nccc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.37
KDM5A P29375 6/20 0.37
KDM4C Q9H3R0 6/20 0.37
KDM5B Q9UGL1 6/20 0.37
NAPRT Q6XQN6 1/20 0.35
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HIF1A Q16665 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
EGLN1 Q9GZT9 2/20 0.34
POLB P06746 2/20 0.34
KDM6B O15054 1/20 0.34
TET3 O43151 1/20 0.34
KDM4A O75164 1/20 0.34
BBOX1 O75936 1/20 0.34
MAPT P10636 1/20 0.34
KDM5C P41229 1/20 0.34
ASPH Q12797 1/20 0.34
KDM4D Q6B0I6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25239224 0.85 PARP1 (0.37) TSHRPOLBMAPTEGLN2SMN1; SMN2
SCHEMBL25237230 0.81 KDM4E (0.40) KDM4CTSHRKDM4EALDH1A1POLB
SCHEMBL31309309 0.72 TPMT (0.39) TTRKDM5AKDM4CKDM5BALOX15
SCHEMBL31114292 0.70 KDM5A (0.33) KDM5AKDM4CKDM5BPIK3CA
SCHEMBL15243426 0.69 HCAR2 (0.41) KDM5AKDM4CKDM5BNAPRTKDM4E
SCHEMBL31114289 0.68 PTGER4 (0.41) KDM5AKDM4CKDM5BMAPTPIK3CA
SCHEMBL15232225 0.68 HCAR2 (0.40) KDM5AKDM4CKDM5BNAPRTKDM4E
SCHEMBL3081703 0.68 ESR1 (0.47) KDM5AKDM4CKDM5BNAPRTKDM4E
SCHEMBL31309518 0.67 ALDH1A1 (0.34) TTRKDM4CALDH1A1POLBKDM4A
SCHEMBL2715907 0.63 DRD2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed