SCHEMBL25254089

SCHEMBL25254089

FC(F)(F)Oc1ccc(-c2nc(Cl)nc3ccccc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.60
ALDH1A1 P00352 3/20 0.60
ACP1 P24666 1/20 0.51
SCN9A Q15858 6/20 0.46
ADORA2A P29274 3/20 0.46
IGF1R P08069 2/20 0.46
LMNA P02545 2/20 0.44
MAPT P10636 1/20 0.44
DHODH Q02127 2/20 0.44
CHRNA7 P36544 2/20 0.42
NUDT1 P36639 2/20 0.41
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25252418 0.81 ACP1 (0.49) ALDH1A1ACP1SCN9AADORA2AIGF1R
SCHEMBL10273110 0.80 SCN9A (0.71) KDM4EALDH1A1SCN9AADORA2A
SCHEMBL17286874 0.80 KDM4E (0.77) KDM4EALDH1A1ADORA2ALMNAMAPT
SCHEMBL808191 0.80 KDM4E (0.77) KDM4EALDH1A1ADORA2ALMNAMAPT
SCHEMBL25257993 0.80 ACP1 (0.48) ACP1SCN9AADORA2ANUDT1
SCHEMBL808420 0.79 KDM4E (0.77) KDM4EALDH1A1ADORA2ALMNAMAPT
SCHEMBL6329397 0.79 KDM4E (0.71) KDM4EALDH1A1SCN9AADORA2ALMNA
SCHEMBL4087331 0.78 KDM4E (0.75) KDM4EALDH1A1ADORA2ALMNAMAPT
SCHEMBL25210790 0.78 CHRNA7 (0.41) KDM4EALDH1A1ACP1DHODHCHRNA7
Hydrochloric Acid SCHEMBL5803147 0.76 KDM4E (0.72) KDM4EALDH1A1ADORA2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250171464-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2025-05-29 US disclosed
US-12275745-B2 Therapeutic compounds and methods of use GENENTECH, INC. (US) 2025-04-15 US disclosed
EP-4436969-A2 BICYCLIC THERAPEUTIC COMPOUNDS AND METHODS OF USE IN THE TREATMENT OF CANCER Genentech, Inc. (US) 2024-10-02 EP disclosed
CN-118451077-A Bicyclic therapeutic compounds and methods for treatment of cancer 基因泰克公司 2024-08-06 CN disclosed
US-20230203062-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-06-29 US disclosed
US-20230203062-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-06-29 US disclosed
US-20230203062-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-06-29 US disclosed
WO-2023097194-A2 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-06-01 WO disclosed
WO-2023097194-A2 THERAPEUTIC COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2023-06-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250171464-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE VHL, TP53, MCL1 KDM4E 2897/4885ALDH1A1 829/4885ACP1 1196/4885
US-20230203062-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE VHL, TP53, MCL1 KDM4E 2897/4885ALDH1A1 829/4885ACP1 1196/4885
US-12275745-B2 Therapeutic compounds and methods of use VHL, TP53, MCL1 KDM4E 2897/4885ALDH1A1 829/4885ACP1 1196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.