SCHEMBL25255599

SCHEMBL25255599

COc1cccc(CNCc2cccc(-n3ccnc3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.54
CYP11B2 P19099 1/20 0.54
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CHRM2 P08172 1/20 0.49
PDE5A O76074 2/20 0.47
TBXAS1 P24557 2/20 0.47
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HTT P42858 1/20 0.46
IDO1 P14902 1/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 2/20 0.46
TP53 P04637 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30245596 1.00 CYP11B1 (0.54) CYP11B1CYP11B2MEN1KMT2ACHRM2
SCHEMBL25425980 0.91 CYP11B1 (0.53) CYP11B1CYP11B2MEN1KMT2ACHRM2
SCHEMBL6389607 0.85 CYP11B1 (0.71) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL29194768 0.80 CYP11B1 (0.51) CYP11B1CYP11B2PDE5ATBXAS1PDE3B
SCHEMBL25426507 0.79 DGAT2 (0.53) MEN1KMT2ACHRM2SMN1; SMN2KDM4E
SCHEMBL30245937 0.79 DGAT2 (0.53) MEN1KMT2ACHRM2SMN1; SMN2KDM4E
SCHEMBL25426299 0.78 CYP11B1 (0.47) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL30245712 0.78 CYP11B1 (0.47) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL25427881 0.78 CYP11B1 (0.46) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL30244976 0.78 CYP11B1 (0.46) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN disclosed
WO-2023018472-A9 AMINOARYL-INTEGRIN AGONISTS COMPOUNDS TEXAS HEART INSTITUTE (US) 2023-07-13 WO disclosed